Ukr. Bioorg. Acta 2020, Vol. 15, N2
hpps://doi.org/10.15407/bioorganica2020.02
CONTENTS
Review article
Olga V. Shablykina, Viktoriia S. Moskvina, Volodymyr P. Khilya
Features of the synthesis and biological evaluation of 3-(carboxyphenyl)chromones
3
Research articles
Stepan G. Pilyo, Оlexandr P. Kozachenko, Victor V. Zhirnov, Maryna V. Kachaeva,
Oleksandr L. Kobzar, Andriy I. Vovk and Volodymyr S. Brovarets
Synthesis and anticancer activity of 5-sulfonyl derivatives of
1,3-oxazole-4-carboxylates
13
Yana I. Sakhno, Maksym V. Mykhailenko, Maksim A. Kolosov, Elena H. Shvets,
Vladimir I. Musatov, Natalia V. Chorna, Sergey M. Desenko and Valentyn A. Chebanov
Condition-based switching the multicomponent reactions of 5-amino-3-(methylthio)-1,2,4-triazole, aromatic aldehydes, and pyruvic acid
22
Anastasiia A. Riabchenko, Olga V. Shablykina, Serhiy V. Shilin, Svitlana A. Chumachenko, Volodymyr P. Khilya
Amino acid sulfonamides based on 4-(1-oxo-1H-isochromen-3-yl)benzenesulfonyl chloride
27
Oleksandr L. Kobzar, Vitaliy O. Sinenko, Yuriy V. Shulha, Vlasyslav M. Buldenko, Diana M. Hodyna, Stepan G. Pilyo, Volodymyr S. Brovarets and Andriy I. Vovk
Synthesis and evaluation of new thiazole-containing rhodanine-3-alkanoic acids as inhibitors of protein tyrosine phosphatases and glutathione S-transferases
33
Anna P. Kryshchyshyn-Dylevych
Some pharmacological properties of 4-[3-(5-bromo-2-hydroxyphenyl)-5-phenyl-3,4-dihydropyrazol-2-yl]-5H-thiazol-2-one
41
Yevheniia S. Velihina, Nataliya V. Obernikhina, Stepan G. Pilyo, Maryna V. Kachaeva, Oleksiy D. Kachkovsky, Volodymyr S. Brovarets
In silico study of binding affinity of nitrogenous bicyclic heterocycles: fragment-to-fragment approach
49